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- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) abstract "Discovery and development of beta-adrenergic receptor antagonists β-adrenergic receptor antagonists (beta-blockers/β-blockers) were initially developed in the 1960s, for the treatment of angina pectoris but are now also used for hypertension, congestive heart failure and certain arrhythmias. In the 1950s, dichloroisoproterenol (DCI) was discovered to be a β-antagonist that blocked the effects of sympathomimetic amines on bronchodilation, uterine relaxation and heart stimulation. Although DCI had no clinical utility, a change in the compound did provide a clinical candidate, pronethalol, which was introduced in 1962.".
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) thumbnail DCI.png?width=300.
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) wikiPageID "41069208".
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) wikiPageRevisionID "597641063".
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) group "Case studies of discovery".
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) group "Steps in design".
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) group "and development of drug classes".
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) list "* ACE inhibitors * Angiotensin receptor blockers * Antiandrogens * Cephalosporins * c-Met inhibitors * Cyclooxygenase 2 inhibitors * Dipeptidyl peptidase-4 inhibitors * Direct thrombin inhibitors * Dual serotonin and norepinephrine reuptake inhibitors * HIV-protease inhibitors * Integrase inhibitors * mTOR inhibitors * Non-nucleoside reverse-transcriptase inhibitors * Nucleoside and nucleotide reverse-transcriptase inhibitors * Proton pump inhibitors * Statins * Thalidomide and its analogs * Triptans * TRPV1 antagonists * Tubulin inhibitors * Bcr-Abl tyrosine-kinase inhibitors * Cannabinoid receptor antagonists * CCR5 receptor antagonists * Neurokinin 1 receptor antagonists * 5-HT3 antagonists * Melatonin receptor agonists * Renin inhibitors".
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) list "* Drug discovery * Drug discovery hit to lead * Drug development".
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) listclass "hlist".
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) name "Drug design".
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) state "autocollapse".
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) title Drug_design.
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) subject Category:Beta_blockers.
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) subject Category:Drug_discovery.
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) comment "Discovery and development of beta-adrenergic receptor antagonists β-adrenergic receptor antagonists (beta-blockers/β-blockers) were initially developed in the 1960s, for the treatment of angina pectoris but are now also used for hypertension, congestive heart failure and certain arrhythmias. In the 1950s, dichloroisoproterenol (DCI) was discovered to be a β-antagonist that blocked the effects of sympathomimetic amines on bronchodilation, uterine relaxation and heart stimulation.".
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) label "Discovery and development of beta-adrenergic receptor antagonists (beta-blockers)".
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) sameAs m.0z8gzfs.
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) sameAs Q17080938.
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) sameAs Q17080938.
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) wasDerivedFrom Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers)?oldid=597641063.
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) depiction DCI.png.
- Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers) isPrimaryTopicOf Discovery_and_development_of_beta-adrenergic_receptor_antagonists_(beta-blockers).