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- Cannabinoid_receptor abstract "Cannabinoid receptors are part of the cannabinoid receptor system in the brain and are involved in a variety of physiological processes including appetite, pain-sensation, mood, and memory. They are also responsible for the mediation of the psychoactive effects of cannabis. Cannabinoid receptors are of a class of cell membrane receptors under the G protein-coupled receptor superfamily. As is typical of G protein-coupled receptors, the cannabinoid receptors contain seven transmembrane spanning domains. Cannabinoid receptors are activated by three major groups of ligands, endocannabinoids (produced by the mammalian body), plant cannabinoids (such as THC, produced by the cannabis plant) and synthetic cannabinoids (such as HU-210). All of the endocannabinoids and plant cannabinoids are lipophilic, such as fat soluble compounds.There are currently two known subtypes of cannabinoid receptors, termed CB1 and CB2. The CB1 receptor is expressed mainly in the brain (central nervous system or "CNS"), but also in the lungs, liver and kidneys. The CB2 receptor is expressed mainly in the immune system and in hematopoietic cells. Mounting evidence suggests that there are novel cannabinoid receptors that is, non-CB1 and non-CB2, which are expressed in endothelial cells and in the CNS. In 2007, the binding of several cannabinoids to a G protein-coupled receptor (GPCR) in the brain was described.The protein sequences of CB1 and CB2 receptors are about 44% similar. When only the transmembrane regions of the receptors are considered, amino acid similarity between the two receptor subtypes is approximately 68%. In addition, minor variations in each receptor have been identified. Cannabinoids bind reversibly and stereo-selectively to the cannabinoid receptors. Subtype selective cannabinoids have been developed which theoretically may have advantages for treatment of certain diseases such as obesity.".
- Cannabinoid_receptor arm "p".
- Cannabinoid_receptor arm "q".
- Cannabinoid_receptor band "14".
- Cannabinoid_receptor chromosome "1".
- Cannabinoid_receptor chromosome "6".
- Cannabinoid_receptor entrezgene "1268".
- Cannabinoid_receptor entrezgene "1269".
- Cannabinoid_receptor hgncid "2159".
- Cannabinoid_receptor hgncid "2160".
- Cannabinoid_receptor locusSupplementaryData "-q15".
- Cannabinoid_receptor omim "114610".
- Cannabinoid_receptor omim "605051".
- Cannabinoid_receptor refseq "NM_001841".
- Cannabinoid_receptor refseq "NM_033181".
- Cannabinoid_receptor symbol "CNR".
- Cannabinoid_receptor symbol "CNR1".
- Cannabinoid_receptor symbol "CNR2".
- Cannabinoid_receptor thumbnail Cb1_cb2_structure.png?width=300.
- Cannabinoid_receptor uniprot "P21554".
- Cannabinoid_receptor uniprot "P34972".
- Cannabinoid_receptor wikiPageExternalLink www.endocannabinoid.net.
- Cannabinoid_receptor wikiPageExternalLink ChapterMenuForward?chapterID=1279.
- Cannabinoid_receptor wikiPageID "586091".
- Cannabinoid_receptor wikiPageRevisionID "604455877".
- Cannabinoid_receptor altsymbols "CNR".
- Cannabinoid_receptor arm "p".
- Cannabinoid_receptor arm "q".
- Cannabinoid_receptor band "14".
- Cannabinoid_receptor caption "NMR solution structure of a peptide mimetic of the fourth cytoplasmic loop of the CB1 cannabinoid receptor based on the coordinates.".
- Cannabinoid_receptor chromosome "1".
- Cannabinoid_receptor chromosome "6".
- Cannabinoid_receptor entrezgene "1268".
- Cannabinoid_receptor entrezgene "1269".
- Cannabinoid_receptor hasPhotoCollection Cannabinoid_receptor.
- Cannabinoid_receptor hgncid "2159".
- Cannabinoid_receptor hgncid "2160".
- Cannabinoid_receptor homologene "1389".
- Cannabinoid_receptor homologene "7273".
- Cannabinoid_receptor locussupplementarydata "-q15".
- Cannabinoid_receptor name Cannabinoid_receptor_type_1.
- Cannabinoid_receptor name Cannabinoid_receptor_type_2.
- Cannabinoid_receptor omim "114610".
- Cannabinoid_receptor omim "605051".
- Cannabinoid_receptor refseq "NM_001841".
- Cannabinoid_receptor refseq "NM_033181".
- Cannabinoid_receptor symbol "CNR1".
- Cannabinoid_receptor symbol "CNR2".
- Cannabinoid_receptor uniprot "P21554".
- Cannabinoid_receptor uniprot "P34972".
- Cannabinoid_receptor subject Category:G_protein_coupled_receptors.
- Cannabinoid_receptor type BodyPart105220461.
- Cannabinoid_receptor type GProteinCoupledReceptors.
- Cannabinoid_receptor type Part109385911.
- Cannabinoid_receptor type PhysicalEntity100001930.
- Cannabinoid_receptor type Receptor105608868.
- Cannabinoid_receptor type Structure105225602.
- Cannabinoid_receptor type Thing100002452.
- Cannabinoid_receptor type Biomolecule.
- Cannabinoid_receptor type Protein.
- Cannabinoid_receptor type ProteinMolecule.
- Cannabinoid_receptor type BiologicalObject.
- Cannabinoid_receptor comment "Cannabinoid receptors are part of the cannabinoid receptor system in the brain and are involved in a variety of physiological processes including appetite, pain-sensation, mood, and memory. They are also responsible for the mediation of the psychoactive effects of cannabis. Cannabinoid receptors are of a class of cell membrane receptors under the G protein-coupled receptor superfamily.".
- Cannabinoid_receptor label "Cannabinoid receptor".
- Cannabinoid_receptor label "Cannabinoïdereceptor".
- Cannabinoid_receptor label "Endocannabinoid-System".
- Cannabinoid_receptor label "Receptor canabinoide".
- Cannabinoid_receptor label "Receptor cannabinoide".
- Cannabinoid_receptor label "Receptory kannabinoidowe".
- Cannabinoid_receptor label "Recettori cannabinoidi".
- Cannabinoid_receptor label "Каннабиноидные рецепторы".
- Cannabinoid_receptor label "مستقبل كانابينويد".
- Cannabinoid_receptor sameAs Endocannabinoid-System.
- Cannabinoid_receptor sameAs Receptor_cannabinoide.
- Cannabinoid_receptor sameAs Recettori_cannabinoidi.
- Cannabinoid_receptor sameAs Cannabinoïdereceptor.
- Cannabinoid_receptor sameAs Receptory_kannabinoidowe.
- Cannabinoid_receptor sameAs Receptor_canabinoide.
- Cannabinoid_receptor sameAs m.02spqz.
- Cannabinoid_receptor sameAs Q421237.
- Cannabinoid_receptor sameAs Q421237.
- Cannabinoid_receptor sameAs Cannabinoid_receptor.
- Cannabinoid_receptor wasDerivedFrom Cannabinoid_receptor?oldid=604455877.
- Cannabinoid_receptor depiction Cb1_cb2_structure.png.
- Cannabinoid_receptor isPrimaryTopicOf Cannabinoid_receptor.
- Cannabinoid_receptor name "cannabinoid receptor 1 (brain)".
- Cannabinoid_receptor name "cannabinoid receptor 2 (macrophage)".