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- Norepinephrine_reuptake_inhibitor abstract "A norepinephrine reuptake inhibitor (NRI, NERI) or adrenergic reuptake inhibitor (ARI), is a type of drug that acts as a reuptake inhibitor for the neurotransmitters norepinephrine (noradrenaline) and epinephrine (adrenaline) by blocking the action of the norepinephrine transporter (NET). This in turn leads to increased extracellular concentrations of norepinephrine and epinephrine and therefore an increase in adrenergic neurotransmission.NRIs are commonly used in the treatment of conditions like ADHD and narcolepsy due to their psychostimulant effects and in obesity due to their appetite suppressant effects. They are also frequently used as antidepressants for the treatment of major depressive disorder, anxiety and panic disorder . Additionally, many drugs of abuse such as cocaine and methylphenidate possess NRI activity, though it is important to mention that NRIs without combined dopamine reuptake inhibitor (DRI) properties are not significantly rewarding and hence are considered to have a negligible abuse potential. However, norepinephrine has been implicated as acting synergistically with dopamine when actions on the two neurotransmitters are combined (e.g., in the case of NDRIs) to produce rewarding effects in psychostimulant drugs of abuse.A meta analysis published in BMJ in 2011 concluded that the selective norepinephrine reuptake inhibitor reboxetine is is indistinguishable from placebo in the treatment of depression. A second review by the European Medicines Agency concluded that reboxetine was significantly more effective than placebo, and that its risk/benefit ratio was positive. The latter review, also examined the efficacy of reboxetine as a function of baseline depression, and concluded that it was effective in severe depression but did not show effects significantly superior to placebo in mild depression.".
- Norepinephrine_reuptake_inhibitor thumbnail Norepinephrine_structure_with_descriptor.svg?width=300.
- Norepinephrine_reuptake_inhibitor wikiPageID "733964".
- Norepinephrine_reuptake_inhibitor wikiPageRevisionID "605995137".
- Norepinephrine_reuptake_inhibitor hasPhotoCollection Norepinephrine_reuptake_inhibitor.
- Norepinephrine_reuptake_inhibitor subject Category:Drugs_acting_on_the_nervous_system.
- Norepinephrine_reuptake_inhibitor subject Category:Monoamine_reuptake_inhibitors.
- Norepinephrine_reuptake_inhibitor subject Category:Norepinephrine_reuptake_inhibitors.
- Norepinephrine_reuptake_inhibitor type Agent114778436.
- Norepinephrine_reuptake_inhibitor type CausalAgent100007347.
- Norepinephrine_reuptake_inhibitor type Drug103247620.
- Norepinephrine_reuptake_inhibitor type DrugsActingOnTheNervousSystem.
- Norepinephrine_reuptake_inhibitor type Inhibitor114724436.
- Norepinephrine_reuptake_inhibitor type Matter100020827.
- Norepinephrine_reuptake_inhibitor type NorepinephrineReuptakeInhibitors.
- Norepinephrine_reuptake_inhibitor type PhysicalEntity100001930.
- Norepinephrine_reuptake_inhibitor type Substance100020090.
- Norepinephrine_reuptake_inhibitor comment "A norepinephrine reuptake inhibitor (NRI, NERI) or adrenergic reuptake inhibitor (ARI), is a type of drug that acts as a reuptake inhibitor for the neurotransmitters norepinephrine (noradrenaline) and epinephrine (adrenaline) by blocking the action of the norepinephrine transporter (NET).".
- Norepinephrine_reuptake_inhibitor label "Inhibidor selectivo de la recaptación de noradrenalina".
- Norepinephrine_reuptake_inhibitor label "NaRI".
- Norepinephrine_reuptake_inhibitor label "Norepinephrine reuptake inhibitor".
- Norepinephrine_reuptake_inhibitor label "Selektiver Noradrenalin-Wiederaufnahmehemmer".
- Norepinephrine_reuptake_inhibitor label "去甲腎上腺素再攝取抑製劑".
- Norepinephrine_reuptake_inhibitor sameAs Selektiver_Noradrenalin-Wiederaufnahmehemmer.
- Norepinephrine_reuptake_inhibitor sameAs Inhibidor_selectivo_de_la_recaptación_de_noradrenalina.
- Norepinephrine_reuptake_inhibitor sameAs NaRI.
- Norepinephrine_reuptake_inhibitor sameAs m.036r9t.
- Norepinephrine_reuptake_inhibitor sameAs Q899668.
- Norepinephrine_reuptake_inhibitor sameAs Q899668.
- Norepinephrine_reuptake_inhibitor sameAs Norepinephrine_reuptake_inhibitor.
- Norepinephrine_reuptake_inhibitor wasDerivedFrom Norepinephrine_reuptake_inhibitor?oldid=605995137.
- Norepinephrine_reuptake_inhibitor depiction Norepinephrine_structure_with_descriptor.svg.
- Norepinephrine_reuptake_inhibitor isPrimaryTopicOf Norepinephrine_reuptake_inhibitor.