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- Orexin_receptor abstract "The orexin receptor (also referred to as the hypocretin receptor) is a G-protein-coupled receptor that binds the neuropeptide hormone orexin. There are two variants, OX1 and OX2, each encoded by a different gene (HCRTR1, HCRTR2).Both orexin receptors exhibit a similar pharmacology - the 2 orexin peptides, orexin-A and orexin-B, bind to both receptors and, in each case, agonist binding results in an increase in intracellular calcium levels. However, orexin-B shows a 10-fold selectivity for orexin receptor type 2, whilst orexin-A is equipotent at both receptors.Several orexin receptor antagonists are in development for potential use in sleep disorders.".
- Orexin_receptor arm "p".
- Orexin_receptor band "11".
- Orexin_receptor band "33".
- Orexin_receptor chromosome "1".
- Orexin_receptor chromosome "6".
- Orexin_receptor entrezgene "3061".
- Orexin_receptor entrezgene "3062".
- Orexin_receptor hgncid "4848".
- Orexin_receptor hgncid "4849".
- Orexin_receptor locusSupplementaryData "-q11".
- Orexin_receptor omim "602392".
- Orexin_receptor omim "602393".
- Orexin_receptor refseq "NM_001525".
- Orexin_receptor refseq "NM_001526".
- Orexin_receptor symbol "HCRTR1".
- Orexin_receptor symbol "HCRTR2".
- Orexin_receptor symbol "Orexin_rec2".
- Orexin_receptor uniprot "O43613".
- Orexin_receptor uniprot "O43614".
- Orexin_receptor wikiPageExternalLink ChapterMenuForward?chapterID=1346.
- Orexin_receptor wikiPageID "13053833".
- Orexin_receptor wikiPageRevisionID "592716442".
- Orexin_receptor arm "p".
- Orexin_receptor band "11".
- Orexin_receptor band "33".
- Orexin_receptor chromosome "1".
- Orexin_receptor chromosome "6".
- Orexin_receptor entrezgene "3061".
- Orexin_receptor entrezgene "3062".
- Orexin_receptor hasPhotoCollection Orexin_receptor.
- Orexin_receptor hgncid "4848".
- Orexin_receptor hgncid "4849".
- Orexin_receptor interpro "IPR004060".
- Orexin_receptor locussupplementarydata "-q11".
- Orexin_receptor name Hypocretin_(orexin)_receptor_1.
- Orexin_receptor name Hypocretin_(orexin)_receptor_2.
- Orexin_receptor name "Orexin receptor type 2".
- Orexin_receptor omim "602392".
- Orexin_receptor omim "602393".
- Orexin_receptor pfam "PF03827".
- Orexin_receptor refseq "NM_001525".
- Orexin_receptor refseq "NM_001526".
- Orexin_receptor symbol "HCRTR1".
- Orexin_receptor symbol "HCRTR2".
- Orexin_receptor symbol "Orexin_rec2".
- Orexin_receptor uniprot "O43613".
- Orexin_receptor uniprot "O43614".
- Orexin_receptor subject Category:G_protein_coupled_receptors.
- Orexin_receptor subject Category:Orexin_antagonists.
- Orexin_receptor subject Category:Protein_families.
- Orexin_receptor type Adversary109773245.
- Orexin_receptor type CausalAgent100007347.
- Orexin_receptor type LivingThing100004258.
- Orexin_receptor type Object100002684.
- Orexin_receptor type OrexinAntagonists.
- Orexin_receptor type Organism100004475.
- Orexin_receptor type Person100007846.
- Orexin_receptor type PhysicalEntity100001930.
- Orexin_receptor type Whole100003553.
- Orexin_receptor type YagoLegalActor.
- Orexin_receptor type YagoLegalActorGeo.
- Orexin_receptor type Biomolecule.
- Orexin_receptor type Protein.
- Orexin_receptor type ProteinMolecule.
- Orexin_receptor type BiologicalObject.
- Orexin_receptor comment "The orexin receptor (also referred to as the hypocretin receptor) is a G-protein-coupled receptor that binds the neuropeptide hormone orexin. There are two variants, OX1 and OX2, each encoded by a different gene (HCRTR1, HCRTR2).Both orexin receptors exhibit a similar pharmacology - the 2 orexin peptides, orexin-A and orexin-B, bind to both receptors and, in each case, agonist binding results in an increase in intracellular calcium levels.".
- Orexin_receptor label "Orexin receptor".
- Orexin_receptor sameAs m.02z4rvk.
- Orexin_receptor sameAs Q7101692.
- Orexin_receptor sameAs Q7101692.
- Orexin_receptor sameAs Orexin_receptor.
- Orexin_receptor wasDerivedFrom Orexin_receptor?oldid=592716442.
- Orexin_receptor isPrimaryTopicOf Orexin_receptor.
- Orexin_receptor name "hypocretin (orexin) receptor 1".
- Orexin_receptor name "hypocretin (orexin) receptor 2".